BopheloLitokisetso

Mikoflyukan: litaelo tsa tšebeliso

foromo litekanyetso li behoa

Ho lokisetsa "Mikoflyukan" thuto eo e bontšitsoeng tlaase mona ka hlahiswa ka mokgwa wa matlapa le concentrations fapaneng ya ntho a sebetsang a kapa ka sebōpeho sa tharollo bakeng sa Infusion. matlapa a soeufetse, potoloha sebopeho le hanyenyane bevelled metshetshe.

Ka matlapa a nang le 50 mg, ea boleng bo le mafolo-folo le ka lehlakoreng la ka ea maikutlo «F», 'me ka ba bang - "50". Letlapeng foromo "Mikoflyukan" 150 mg, ea a sebetsang a motsoako o - «F150» le mola fihla moo ho arohanang, ka ho latellana.

Ho lokisetsa tharollo ke colorless, e pepeneneng, ntle le likaroloana efe kapa efe.

Sebopeho: Tablets

Active ntho: fluconazole - 50/150 mg, (1 tab ya.).

Excipients:

- ka silicon dioxide e ,

- lactose,

- povidone,

- magnesium stearate

- Valium,

- talc,

- selulose mikrokristallicheskayae

tharollo

Active ntho: fluconazole - 2/200 mg, (1 ML vial le 1, ka ho latellana).

Excipients:

- Metsi bakeng sa ente,

- sodium chloride.

The bohato diokobatsi ya moriana "Mikoflyukan"

Tataiso e bolela hore ho lokisetsa ho amana le mahlahana antifungal tsa sehlahisoa triazole. Fluconazole thibela metsoako ergosterol tswakana tjena: e fana ka e lumellang metsi ho kena ea leboteng ka seleng. Lithethefatsi sebetsang khahlanong Microsporum, Candida, Trichophyton, Cryptococcus neoformans.

Tšobotsi e 'ngoe ea ho bohato diokobatsi ya moriana ke hore ke bobeli khetha sesitisa tsa cytochrome P450 ka li-fungus, empa ka nako e tšoanang, ha e bontša mosebetsi ofe kapa ofe khahlanong le tsamaiso ena e potlakisang tsebetso ea lik'hemik'hale ho batho.

Pharmacokinetics

moriana o hantle-ananelang ka mor'a tsamaiso, 'me ja lijo hammoho le ho nka lithethefatsi ha ho ame absorption lona. Bioavailability - 90%. lithethefatsi e ajoang ho makala ohle le lisele tsa 'mele. Ka tsela eo ea mahloriso ea eona e leng lero la mali mahloriso lekana le makala a latelang le lisele: kopanetsoeng mokelikeli, lebese, mathe, maro ka bosaling, sekhohlela le mokelikeli perinatal, le cerebrospinal mokelikeli bioavailability ka Range ho tloha 50 ho ea ho 90%.

Ho feta moo, litho tsa ka hare tse ling le lisele tsa mahloriso lithethefatsi ka 'na feta ea mahloriso ka lero la mali e. Har'a bona, ho epidermis, ho dermis, ho stratum corneum, fufuleloa mokelikeli. The halofo bophelo - ka 30 lihora tse.

Bontšang bakeng sa tshebediso ya lithethefatsi "Mikoflyukan"

Thupelo ea bolela hore lithethefatsi e na le mosebetsi le phahameng khahlanong le microorganisms tsa mafu tse latelang, tse le tsekamelo ea ho tšoaetsoa mafu fungal:

  • systemic candidiasis,

  • cryptococcosis,

  • mucosal candidiasis,

  • bosaling candidiasis,

  • thibelo ea tšoaetso ea fungal

  • mycoses letlalo,

  • onychomycosis,

  • pityriasis versicolor,

  • parakoktsidiovikoz,

  • coccidioidomycosis,

  • pistoplazmyuoz,

  • sporotrichosis.

Lehlakoreng liphello tsa moriana "Mikoflyukan"

Reviews of sehlopha teko mor'a letoto la lithuto tsa lithethefatsi, ho akarelletsa le placebo-teko le mekhoa e meng ea ho etsa lipatlisiso li bontšitse hore lithethefatsi ka 'na ba tse latelang litla-morao:

- mabapi le pampitšana tshilong ya dijo:

  • bohloko mpeng,

  • ho nyekoa ke pelo,

  • flatulence,

  • letšollo;

- mabapi le bohareng makala tsamaiso ea methapo:

  • ho tsekela,

  • hlooho;

- mabapi le kulisa:

  • liphetoho anaphylactic ea phelang,

  • letlalo lekhopho.

Contraindications ho moriana "Mikoflyukan"

Litaelo ho moriana o bolela hore contraindications ho baeti ba fihlelang ho sona e nyenyane ka ho lekaneng, har'a bona:

  • ho fihlela ho 1 selemo,

  • ea bokhachane,

  • nahanela ho komponeng triazole le fluconazole.

ditshebeditsano lithethefatsi

Prothrombin nako eketseha ha tšebeliso ea lithethefatsi anticoagulant coumarin mofuta.

Derivatives tsa sulfonylurea mahlahana molomo hypoglycemic haholo eketsa bona halofo ea bophelo ba ka kopana le fluconazole.

Fluconazole halofo bophelo nakong e fokotsehile ha ikopanya le rifampicin.

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