Bophelo, Litokisetso
Lithethefatsi "Buspirone": ulasan pelanggan lingaka
hore na ba sebelisa lithethefatsi kapa ho molemo "Buspirone"? Guest, ea neng a sesebelisoa sena tla tšohloa mona ka tlase. Re boetse re u bolella ka seo thepa ya Maemong a itse lithethefatsi eo a neng a e behiloeng, haeba a ena le contraindications efe kapa efe le litla-morao.
Sebopeho le ho hlophisoa ha moriana
Seo ke karolo ea "buspirone" lithethefatsi? Reviews of lingaka re dintho joalo a sebetsang a kang buspirone hydrochloride. Ho phaella moo, moriana o na le metsoako e ka ho eketsehileng ka mokgwa wa lactose, starch poone, k'halsiamo hydrogen phosphate dihydrate, starch (mofuta A), sodium, colloidal silicon e dioxide, magnesium stearate le MCC.
Fumaneha ke sesebelisoa ka mokgwa wa e tšoeu, matlapa a potoloha kenngoa ka e le qubu ea lebokoso.
The pharmacodynamic thepa ya moriana
Seo thepa ea meriana "Buspirone"? Litaelo, maikutlo lingaka tsebisa bakuli ka seo ke anxiolytic lithethefatsi. E ne a rerile hore ho phekola mafu a ho matšoenyeho a simolohile tse sa tšoaneng.
The mochine e tobileng ea bohato matlapa e sa hlomamisoa. Leha ho le joalo, litsebi li pheha khang ea hore lithethefatsi ke khetha agonist ka postsynaptic receptors 5-HT 1a tsamaisong ea methapo ea kutlo.
Ka mor'a ho nka lithethefatsi butle-butle bontša ketso lona. e le hantle ho ka bonoa ka libeke tse 'ngoe ho tse peli. The lebetsoeng le phekolo e le hantle o ne a ile a re feela ka mor'a hore ka khoeli.
The pharmacokinetic thepa ya moriana
Moo absorption ea lithethefatsi "Buspirone"? litsebi Guest fana ka maikutlo a hore lithethefatsi ena haholo ka potlako le hoo e ka bang ka ho feletseng ananelang pampitšaneng gastrointestinal. Ea mahloriso lero la mali lithethefatsi o ile a re ka mor'a lihora tse 1-1.5. Ho buisana le liprotheine e 95% le halofo bophelo - lihora tse tharo.
Hoo e ka bang 30-65% ea chesehang ea mafolofolo motsoako o le metabolites lona di excreted ka moroto le motšehare 'me 20-40% di behilwe hammoho mantle ena. Ha mokuli a na le mathata a le sebete 'me liphio ho felisoa bona decreases hanyenyane.
Ho bonahala lebaka la ho sebelisa matlapa
Ka morero ofe ka lithethefatsi tse kang "Buspirone" ka behilweng? Reviews of lingaka re lithethefatsi ena e sebelisoa ka ho ba teng ha mafu a ho tšoenyeha hore ba tsamaea le matšoao a kang ho imeloa kelellong, ho tšoenyeha le eketsehile ka makhetlo ho tšoenyeha.
Contraindications ho tšebeliso ea lithethefatsi le
Eng ka boemo ba mokuli e thibetsoe ho noa meriana "Buspirone"? litsebi Guest re lithethefatsi ha baa lokela ho e beuweng ho batho ba nang le hypersensitivity tsa motheo le tlatsetso dintho lithethefatsi, myasthenia gravis, a hlobaetsang le congestive glaucoma, matla renal kholofalo, sethoathoa le ho matla ho se sebetse sebete.
Ho feta moo, nahana ka lithethefatsi e contraindicated ka bana ba le nakong ea kanyeso.
Lithethefatsi "Buspirone": litaelo tsa tšebeliso
Maikutlo ka moriana ona o tla hlahisa e nyenyane ho feta.
The Melawana hapa ho moriana o le e tlaleha hore lethal dose lokela ho khetha feela ke ngaka ho ba teng, ho itšetlehile ka boemo ba mokuli.
Hangata, qalong ea kalafo lithethefatsi o laolwa ka ka tjhelete e ya milligrams hlano makhetlo a mararo ka letsatsi. Reng o butle-butle eketsa lethal dose ho 15-30 mg, (partitioned ka tekanyetso 'maloa).
The lebetsoeng le letsatsi litekanyetso li behoa ea ea lithethefatsi ha ea lokela ho ba ho feta 45 mg,, 'me le' ngoe - ha ho ho feta 30 mg,.
Ke lokela ho nka "Buspirone"? Thupelo ea bolela hore a etelle pele lipilisi e lokela ho ba letsatsi le letsatsi ka nako e tšoanang. Ba ke ke ba hlafuna. Lithethefatsi lokela ho feela noa e nyenyane ea metsi.
Batho ba nang le a liphio mosebetsi phytoteratology kapa sebete lokelang ho khoneha litekanyetso li behoa tlaase-tlaase.
Nako Ke 'nete hore e ikemiselitse ka bomong (a sebetsa nyeoe ea ka nyeoe e' ngoe). Ho e hanetsoeng ho nka lithethefatsi bakeng sa nako e telele, haholo-holo ka ntle ho tataiso ea meriana.
Ka e tšoanang le kalafo kgothaletswa sotsioterapevticheskie me litekanyo psychotherapeutic.
maemo a ho overdose
Seo ba lipontšo tsa overdose etsahala ha nka tekanyetso e phahameng ea lithethefatsi "Buspirone"? litsebi Guest fana ka maikutlo a mefuta e latelang: cramps, ho nyekoa ke pelo, mokhathala, molikoalikoane, ho tšitiso ea mala, ho hlatsa.
Ka overdose gastric lavage e entseng, hammoho le go baya leitlho ea khatello ea mali, respiration, le ho otla ha pelo. Kalafo - bontshang matshwao.
litla-morao
Na litla-morao tsa lithethefatsi "Buspirone Sandoz?" Reviews ba bakuli le lingaka li bontša hore lithethefatsi e ka etsa hore ba bangata e khōlō ea liketsahalo e bohloko:
- myocardial infarction, tahlehelo ea nakoana ea kelo-hloko, ha pelo, bao e seng e itseng sefubeng bohloko, setorouku, tachycardia, bradycardia, hypotension kapa kgatelelo ya madi, cardiomyopathy;
- conjunctivitis, thothofatsang pono, boikutlo ba khatello ea ka mahlo, redness ea lihaha-'mele, bohloko boikutlo ka mahlong, narrowing tšimo ea pono, ho hlohlona, photophobia;
- teneha, ho tšoenyeha phytoteratology tšebelisano, litoro tse tšosang, mafu extrapyramidal, lefu la ho hlobaela, ho sisinyeha ho itlelang feela, ho tšoha, ha thothomela hohle, thabo, likhathatso tsa molumo, bora, khopolong ea phytoteratology, ho tepella maikutlo, lipuo slurred, ho otsela, lefu serotonin, molikoalikoane, ho shoohlo, fokotseha hloko, stupor, pherekano, feto-fetoha, depersonalisation, agoraphobia, molumo oa nahanela, feberu, hyperkinesia, phytoteratology amanang ka temoho, ho iphapanya ha batho, nyakallo, gallyutsi se seng, ho ipolaea hylophobia, paresthesia, sethoathoa, lefu Parkinson, boemong bo sa thabiseng, lethargy, psychosis, akathisia;
- kgafetsa ho ntša metsi, mosese tshegetsa le go tlotla, bosiu ho ntša metsi, enuresis;
- epistaxis, nasal tsubuhlellano, bokhutšoanyane phefumoloho, 'metso, bokhutšoanyane phefumoloho, khutsufatso ea pelo;
- arthralgia, ho satalla le mesifa spasm, myasthenia, myalgia;
- liphetoho entsprechen mali;
- batang hypersensitivity, mokhathala, tšekamelo ea ho noa ka tsela e feteletseng ea joala, ho tšoaroa ke hlooho, phytoteratology mali hoama, eketsa kapa fokotseha ka boima ba 'mele, le chesang mahlaseli, boikutlo ba ho ba ringing ka hlooho, lekhopho, malaise, mokhathala, phytoteratology tatso le monko, tahlehelo ea lentsoe, hiccups, glossalgia;
- tinnitus;
- mafu matsatsing, fokotseha kapa eketsehileng libido, ho ruruha ya urogenital makala, amenorrhea, ho hloka matla, fokotswa ntsha peo;
- lekhopho, edema, ecchymosis, hyperemia, pemphigus, alopecia, e omeletseng, eczema, kulisa, urticaria, thinning ea Nail, hematoma;
- letšollo, ho teneha feela mantle a syndrome,, salivation, ho nyekoa ke pelo, ho tebelwa mosebetsing ea mali ho tswa rectum e, epigastric bohloko, phahameng sebete enzyme, molomo o omileng, pipitlelano, flatulence, e ile ea eketseha kapa fokotseha maikutlo a tlala, ho hlatsa;
- galactorrhea, phytoteratology thyroid mosebetsi, gynecomastia.
ditshebeditsano lithethefatsi
Pele o sebedisa "Buspirone" lithethefatsi lokela ho ba bonnete ba hore bala ditaelo. Ho fana ka boitsebiso bo latelang ka ditshebeditsano lithethefatsi boletsweng lithethefatsi:
- Ha ho kopantswe le antidepressant e, antihypertensive mahlahana, glycosides cardiac, anticoagulants, hypoglycemic le mahlahana neuroleptic hammoho le lithibela-pelehi molomo hloka ka tieo taolo ea meriana. Sebelisana le sedatives le benzodiazepines sa amoheleheng.
- inhibitors e matla ea cytochrome P450 keketseho e bioavailability "buspirone".
- E sa kgothaletswa ho nka lithethefatsi le Mao inhibitors ka lebaka la ketsahalo e sa khoneha sa bothata hypertension.
- Hammoho le kenoa "Cimetidine" palo e kahodimodimo ea mahloriso "buspirone Sandoz" e ile ea eketseha ka 40%.
- "Rifampicin" fokotsa palo e kahodimodimo ea lithethefatsi mahloriso ka bang 89,6%.
- Ha ho kopantswe le lithethefatsi tse amang ea mahloriso palo e kahodimodimo ea "buspirone", ke tse lakatsehang ho fetola ho lethal dose ea bobeli.
- "Ritonavir" le "ketoconazole" le literata le tsa likokoana-hloko phetoho "buspirone" hammoho le eketsa lero la mali mahloriso lona.
- Le ha e kopana le ea lithethefatsi e le "diazepam" dikahare tsa bobeli ka e ile ea eketseha ka lero la mali mali. Ho phaella moo, ho ka ba le litla-morao tse kang ho nyekeloa ke pelo, ho tsekela 'me hlooho.
- Tsoa hong ho amohelloang "buspirone" le "Haloperidol" a ka eketsa maemo le serum.
- Ho lokela ho qoba ho noa joala ka nako kalafo "buspirone Sandoz."
Lithethefatsi "Buspirone": Testimonials tsa batho (bareki) le litsebi
bakuli fetisisa siea poeletsotlaleho ntle ka lithethefatsi ena. Ba ela hloko bokgoni lona phahameng. About litla-morao e ile ea tlaleha ka seoelo haholo.
Litsebi li bolela hore ho nka lipilisi tsena hase hangata haholo etsa hore liphello tse sa rateheng. Ba ka feela ho ketekoa ka sehlopha fapaneng tsa bakuli. Tabeng ena, litla-morao tse bonolo feela 'me ka potlako feta ntle discontinuation ya moriana.
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