Bophelo, Litokisetso
Drotaverina hydrochloride
hydrochloride Drotaverina amana hlophisitsoeng meriana le phello e spasmolytic. mosebetsi lona e lebisitsoe ho mesifa le boreleli la tshilong ya dijo makala, urogenital le biliary tsamaiso, hammoho le vascular boreleli mesifa lera. Drotaverina hydrochloride (Nospanum), ho kgothaletsa boikhathollo tsa le dikarolo boreleli mesifa, o tla khona ho felisa cramping. Ho feta moo, lithethefatsi ntlafatsa dinama tse nyenyane tse phepo e ntle oksijene ka ho atolosa vascular lumen. Drotaverina hydrochloride na le matla a ho fetola ea bokgoni ba lera sele le e lumellang metsi ho kena. The moriana o fokotsa mosebetsi enzymatic tsa phosphodiesterase, khothalletsa batho ka tsela e lumellanang (junifomo) eketsa Camp maemo le absorption ea pele ea lisele tse k'halsiamo Ion.
Drotaverina hydrochloride tšoauoa ka tsela e itseng e tlase ya coupling le liprotheine lero la mali. Hangata e tlama ho tsa beta le Alpha-globulin, albumin. Mor'a metsotso mashome a mane a metso e mehlano le mashome a tšeletseng ka mor'a tsamaiso molomo le lero la mali kopo bontša mahloriso tlhōrō ea ntho mafolofolo. The halofo bophelo ba ka taelo ea lihora tse mashome a mabeli a metso e 'meli. Excretion tsa metabolites hlahiswa haholo-holo ka moroto wa. Karolo ea excretion ea moriana o hlahellang teng masi le.
Moriana o (ka sebōpeho sa ente e, 'me matlapa a) abetsoe ho felisa bohloko boo se bo le spastic tlhaku cupping spasm. hydrochloride Drotaverina bontša gastric seso, cholecystitis, pipitlelano, spastic etiology, pyloric boreleli mesifa spasm le mok'hadinale gastric karete, cystitis, nephrolithiasis, proctitis, pyelitis le uretrolitiaze. Lithethefatsi e sebelisoa ka cramps mala bakoang ke likhase lieha le spastic colitis. moriana o le ka boela sebelisoa ha re khanna tlhathoba, ho akarelletsa le holetsistografii ena. Drotaverine abeloa ho vasodilatation ka boitsebahatso ea vascular mesifa boreleli spasms lera remover hlooho spasm ea methapo ea bokong. moriana o sebelisoang hangata ka algodismenoree ikatisetsa gynecological. The moriana o ke khona ho thibela le ho felisa mesifa boreleli cramps ka popelo ka nakong ea bokhachane 'me tabeng ea soka ho ntša mpa. E boetse e bontša ka nako pelehi bakeng sa spasmolysis le bo tsoelang pele tsebagatswe uterine metso 'me ka linako postnatal.
Drotaverina hydrochloride. Litaelo.
ho lokisetsa e ka mokgwa wa matlapa ea lokela ho nkoa ka molomo. Tablets ha baa lokela ho hore di hlafunnwe kapa e sithabetseng, e lokela ho metsoa kaofela, ka metsi ka bongata bo lekaneng. Lithethefatsi ha ea itšetleha ka nako ea lijo. The litekanyetso li behoa 'me nako ea phekolo o ikemiselitse ka bomong ke ngaka ho ba teng.
Bakeng sa bacha (ba fetang leshome le metso e lilemo tse) le batho ba baholo ho imolla mahlaba spastic thonya matlapa 1-2 (40-80 mg,) ka makhetlo a mabeli kapa a mararo ka letsatsi.
Bana ba ka tlaase lilemo tse leshome le metso e ea ho lokisetsa o fuoa ho ea ka ho khethoa ha ho ngaka.
The moriana o ka sebōpeho sa ente e laolwa intramuscularly. Bakeng sa bakuli ba insufficiency renal kapa e amanang le sebete, e ka fokotsa ho qaloa ho moriana entoe. Joalo mokhoa o utloahalang a feela ka mor'a hore ho nkeloa ka lapeng la boemo tshekaletseng tsa mokuli. Ka pheriferale ho potoloha ha mali pherekano e bakoang ke vascular boreleli mesifa spasm lera ho lieha intraarterial tsamaiso.
E le busa, bakuli ba a mamella meriana. Leha ho le joalo, maemong a mang, ho ka ba le litla-morao. Mohlala, bakuli ba ka 'na ba ho nyekeloa ke pelo, nang le bokooa setuloana, ho hlatsa. Ka 'na etsahala,' me CNS mafu a, tse kang tlōlo ea falimehe le mokgwa wa ba bang kaofela (ho robala), hlooho e opang, fainting. Ho ne ho maemo a ho lefu la ea tsamaiso la pelo, o ile a bontša ka ho tachycardia, arrhythmias, theola khatello ea. Hape, hoa khoneha ho ruruha ya nasal mucosa, kulisa, bronchospasm.
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