Bophelo, Litokisetso
"Bisoprolol": litaelo tsa tšebeliso
Ho lokisetsa "bisoprolol-Praana" ke matlapa a 10-milligram, tse a tlotsitsoeng kenapa lijo. Letlapa e mong oa lithethefatsi ena e na le 5, mg bisoprolol fumarate, e leng ba ka sehloohong a sebetsang a ntho.
Ntle ho, ba thusang, ea moriana o kenyelletsa ditokiseletso primellozu, povidone, starch, aerosil, talc, microcrystalline selulose, magnesium stearate. Tablets shell dikarolo di polyvinyl joala, thaethaniamo dioxide, colouring oxide e tšepe, talc, macrogol.
Sebediswa ho dipakete 30 Letlapa.
The bohato diokobatsi ea lithethefatsi "bisoprolol" taeo pukwanana hlalosang ka tsela ena. lithethefatsi ena e na le thepa, eo netefatsa antianginal, antiarrhythmic, hammoho le e atlehang hypotensive bohato. Ka lebaka leo, ho bonahala ka sehloohong bakeng sa ho e sebelisa reretsoe ke mafu a kang kgatelelo ya madi le mefuta e sa tšoaneng ea arrhythmia, angina pectoris. E le e atlehang ho phekola lithethefatsi sebediswa bakeng sa kalafo le thibelo ea ho hloleha itekanetseng pelo le myocardial nako.
Contraindications ho tshebediso ya moriana o ba hypersensitivity mamello ho dikarolo tsa moriana, fumanoa sinus bradycardia, cardiogenic makala, cardiac le ho hloleha ho hema tseleng e mpe ea ho kula. Ho sebelisoa ha lithethefatsi nakong ea bokhachane le nako diabolololo lokela ho latela ka tekanyo e oa ka monyetla oa likotsi hlahang ho tloha e sebelisa. Ho seng joalo, e ne e ka sokela ho ntshetsopele ya tlhaka bao e seng congenital kapa ngoana. Haeba meriana e etsoa ka nako ea mosali ka matsatsi a tlase ho tse peli tse kapa tse tharo pele ho fana ka puo, na e lokela ho ba e khethehileng ya kalafi go baya leitlho ya lesea.
Lithethefatsi "bisoprolol" Taeo ka kopo e khothalletsa ho noa ha mokelikeli, hangata hoseng pele u ja kapa nakong ea lijo tsa hoseng, ho hlatsoa ho theosa le lipilisi u hloka e nyenyane ea metsi. The lethal dose ea letsatsi le letsatsi ea tsamaiso ea lithethefatsi le 'ngoe e 1,25-10 mg,. Haeba ho hlokahala, lethal dose ea ka e ile ea eketseha, empa feela ka go baya leitlho ea kamehla ea ho otla ha pelo ea mokuli le ho hatelloa.
Ho itšetlehile ka mofuta oa boloetse fapana lithethefatsi tsamaiso lethal dose. Kahoo, ha e le e lekanang kgatelelo ya madi 5,10 mg,, 1,25 mg, - sa foleng ho hloleha. Kalafo o etsoang tsoa ka matsatsi a supileng. Ka mamello ho tloaelehile ho kalafo ya ea lithethefatsi e tsoela pele ho latela sekemeng, e leng e hlalosa ka ho qaqileng ka litaelo tsa ho sebelisa mehaho ea moriana. Leha ho le joalo, e lokela ho utloisisa hore ho lethal dose palo e kahodimodimo ea lithethefatsi ka ho ya ka letsatsi le ka 'na sa feteng 20 milligrams.
Ka ho lokisetsa "bisoprolol" taeo pukwanana e bua ka tse latelang litla khoneha lehlakoreng. E lokela ho jere hopola hore poleloana e reng bona, tse ngotsweng ditaelo, e sebetsa feela ho mabokosana moo lethal dose ea meriana e sa feteng 40 milligrams.
Ditlamorao tsa hlokomela le litsamaiso tse sa tšoaneng tsa 'mele, ho etsa mohlala, ea tsamaiso ea methapo ke ho tsekela, ho tepella maikutlo, ho tšoenyeha, ka seoelo - lipono le ho nahana ho hloka taolo, bonwang ho hloka taolo.
Ka lehlakoreng la pampitšana tshilong ya dijo ke liketsahalo o tloaelehileng haholo oa letšollo, ho nyekoa ke pelo, dyspepsia fapaneng. Khoneha lekhopho, kulisa ka letlalo, dermatitis. Ka kalafo lithethefatsi, "bisoprolol" taeo ka kopo e bontša ka monyetla oa ho ba ketsahalo e ea ho tšoaroa ke hlooho le ho utloa bohloko bo tšimong ea epistragalnoy, involuntary keketseho ea boima ba 'mele.
sebelisana lithethefatsi ho lokisetsa e tšoauoa ka tsela e latelang. Haeba u noa meriana "bisoprolol" le amiodarone, verapamil, alpha methyldopa, quinidine meriana, moo ho na le ke kotsi ya ditlolo tsa automaticity le contractility eketseha pelo. Tsamaisana lithethefatsi le Mao inhibitors.
Ka overdose kgothaletswa gastric lavage, kena le mamello adsorbing lithethefatsi (atropine), sedatives le mahlahana cardiotonic (epinephrine, diazepam, lorazepam, joalo-joalo), And glycosides cardiac. Tabeng ea le literata pelo ka potlako ho hlokahala transvenous tlhotlheletso.
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