BopheloLitokisetso

Seo "Piracetam" nka? Litaelo tsa tšebeliso "piracetam"

Seo "Piracetam" balletsweng bakuli? The karabo ea potso ena, u tla ithuta ho tloha sehlooho sena. Hape, re tla nehelana ka uena ka boitsebiso bo mabapi le kamoo ho nka pheko ena, eo ho eona theha e le teng, hore na litla-morao 'me contraindications, ka sebelisoa nakong diabolololo le ho ima.

ho lokolloa foromo ea lithethefatsi, ambalaji le sebopeho

Pele re u bolella ka seo "Piracetam" e balletsweng ke ngaka lokela bolella ka seo theha e ka rekoa ka na bapharmasi.

Kajeno, ho na le liforomo tse 'maloa tsa ea lithethefatsi ena. A re ke re tšohleng lipotso tseo ka ho qaqileng le ho feta.

  • Capsules. mofuta ona oa moriana o na le 0,4 g, piracetam le marketed ka lebokoso dipakete likotoana tse 60.
  • 20% tharollo. foromo ena e rekiswa ho ampoules 5 di ml ka seng, e leng, le eena, a kenngoa ka mabokose a likotoana 10.
  • Tablets. Lithethefatsi-a tlotsitsoeng mosehla 'me e na le 0,2 g ya ntho mafolofolo. Tablets a ka fumana ka lebokoso sosobaneng ke likotoana 120 kapa tse 60.
  • Granules bakeng sa bana. Lithethefatsi na leseli pinki mmala (re brownish pellet), e fumaneha ka linkho khalase bakeng sa '56

E lokela ho ile a hlokomela hore e mong le mofuta o mong oa lithethefatsi o na le excipients lona.

Pharmacodynamics moriana o

Seo "Piracetam" ka fuoa kabelo ea ho motho? Ena lithethefatsi nootropic eo o khona ho fana ka le phello e ntle ka ajoa boko le metabolism.

The moriana o ntlafatsa dithulaganyo tshilong ya dijo le kgothaletsa tsoekere tshebediso. Hape, ho thibela aggregation tsa liplatelete butswe.

Baeti ba fihlelang ho "piracetam" e na le phello sireletsang diso boko hore li bakoa ke motlakase makala, botahoa, kapa hypoxia. Ho feta moo, lithethefatsi ena ntlafatsa integrative boko mosebetsi ntle ikitlaetsa psychostimulant le robatseng.

The thepa ya moriana

Seo thepa ya lithethefatsi "Piracetam"? Seo e balletsweng ke ho bolela? O ne a nka lithethefatsi kgona ho ebe o kenya tshebetsong dithulaganyo amanang ka ka CNS, hammoho le ho ntlafatsa feto-fetoha le memoring ya ka bakuli ba ka le ho bafo ba phetse hantle.

Seo "Piracetam" ka abeloa ho ea bana? sesebelisoa sena ke khona ho eketsa mosebetsi kelello, ho ntlafatsa tshebetso a kelello, bebofatsa dithulaganyo ithuta, ho ntlafatsa conductivity (synaptic) ka cortex bokong le puisano pakeng tsa hemispheres lona (setseng le letona). lithethefatsi tsosolosa le ho tsitsisa le litsebeng puo, karete ya memori le kelo-hloko.

Molao-motheo oa ketso ea lithethefatsi ka

Joang lithethefatsi "Piracetam"? Bakeng sa seo e se e sebediswa bakeng sa bacha le batho ba hōlileng?

Ba ne ba nka ho lokisetsa normalizes karo-karolelano ea ATP le ADP, 'me hape activates phospholipase A, eketsa le ntsetso-peleng le phapanyetsano ya polasetiki neurotransmitter tlhotlheletso le dithulaganyo bioenergetic ka lisele tšohile.

Seo "Pyracetam" (liente, phofo, capsules le matlapa) ka laolwa bakuli? lithethefatsi Sena se ka thibela platelet aggregation, ntlafatsa microcirculation le optimize tshebetso ya ho feta erythrocytes ka lijaneng tse nyenyane.

Hape re lokela ho ela hloko hore thulusi ena eketsa lebatowa ajoa mali libakeng tse ischemic ea boko, ho matlafatsa, alpha le tsa beta mosebetsi, empa ka nako e tšoanang ho fokotsa mosebetsi oa noka.

Meriana ho fokotsa skeletal nystagmus. Nakong hypoxia, ho sithabela le botahoa o na le litla neuroprotective.

Mabapi le thepa-ba khahlanong le hypoxic ea lithethefatsi a sebetsang a ke haholo e atlehang ea ho phekola ba infarction myocardial.

Pharmacokinetics ya moriana

nako e kae meriana e ananelang "Piracetam" (e leng se bolelang hore e abetsoeng, re tla bolella hamorao)? Ka mor'a tsamaiso molomo lithethefatsi ka potlako le ka ho feletseng ananelang. bioavailability lona ke ba etsang liphesente tse lekholo.

tsamaiso molomo ya moriana o ka tjhelete e ya 2 g, a fana ka mahloriso lebetsoeng le ka lero la mali ka mor'a metsotso e mashome a mararo. E Bolela ha tlama ho liprotheine tse phunyeletse makala ohle le lisele, ho akarelletsa le placenta ho.

Meriana hoo e batlang e ha metabolized, 'me khetha bakoang ka parietal, occipital le tse tobileng libakeng tsa boko, hammoho le ka cerebellum le basal ganglia.

The halofo bophelo ba lisebelisoa ke lihora tse hlano. About 95% ya lithethefatsi excreted ka moroto le foromo e sa fetohe (ka mor'a ka mashome a mararo lihora tse). Ka batho ba nang le renal ho hloleha fanoeng eketseha nako.

Ke hobane'ng ha re hloka "Piracetam"? ho bonahala

Nkoa nootropic moemeli o na le a manyenyane sephara ea khato. Ho ea ka litaelo tseo, ka bontšang bakeng sa ho e sebelisa ke re lintho tse latelang:

  • ischemic leqeba le liphello tsa lona;
  • cerebrovascular insufficiency foleng mofuta (mohlala, arteriosclerosis, hypertension vascular lefu kapa Parkinson), a tsamaea le ho tšoaroa ke hlooho, molikoalikoane, ho kholofalo memori, tlhokomelo le ho bua;

  • dementia '(ho akarelletsa le lefu la Alzheimer);
  • aphasia;
  • neuroinfection bongata ba kokwanahloko (a hlobaetsang le);
  • mafu a ea tsamaiso ea methapo ea kutlo, a tsamaea le ea fokotseha ka mesebetsi ea kelello le mnemonic, tekanyo ea ho falimehe, hammoho le khahlanong le boitšoaro bo ka maikutlo le volitional;
  • botahoa (ho akarelletsa le nako ea ho hlaphoheloa, subkomatoznoe le coma) ;
  • ho tsekela;
  • tsehetso ea hlabollo-manyolo mafu a;
  • noabolohang le thahaselle mmuso;
  • cortical myoclonus;
  • sithabetsang boko ntsa kotsi;
  • sethoathoa (jwalo ka adjuvant e);
  • skeletal nystagmus;
  • le senile atrophic dithulaganyo.

Ha bopengwi efe kapa efe ntse ho laela lithethefatsi "Piracetam"? Hobaneng noa ho bolela le ho etsa liente? , Ho phaella ho ka holimo, lithethefatsi ena e na le bopaki bo kang:

  • methapo ea kutlo, somatovegetativnye, mathata a mafu a kelello ka mor'a kalafo le lithethefatsi psychotropic le antipsychotics;
  • hlobaetsang botahoa le se entsoeng ka amphetamine, ethanol, barbiturates kapa morphine e;
  • ho tepella maikutlo manganga ho kalafo antidepressant;
  • neurotic ho tepella maikutlo le asthenia le maloetse a senesto-hypochondriacal, hammoho le, 'me liketsahalo adynamia ideomotor thibelo;
  • khaotsa ho tsuba, pele - le e re delirious ka bokhoba ba tahi le ho lemalla lithethefatsi;
  • tsehetso ea hlabollo-manyolo lefu ka ho lemalla joala (sa foleng);
  • sekele khaello ea mali a ka cell (ka kalafo).

Seo "Piracetam" matlapa a le capsules le phofo, lingaka hangata e buella ho fumana bakuli ba bona ba banyenyane? ho lokisetsa e joalo e ba laela hore bokong palsy kholofalo kelellong, liphello tsa perinatal CNS, tlaase ho ithuta (ha psychoorganic lefu), kholofalo kelellong, mafu a lipuo le kholofalo hopola insufficiency kelello.

Diabolololo le ho ima

Nka nka lithethefatsi "Piracetam" nakong ea bokhachane? Ho etsa? Litsebi tse ling li laela ho nkoa le mokhoa oa ho basali le boemong ba ho bontša. Leha ho le joalo, e lokela ho hopola hore lithethefatsi habonolo lifapano le mokoallo placental le ka lebese. Tabeng ena, e contraindicated nakong diabolololo le emara. Ho seng joalo, e ne e ka ba kotsi ho bophelo bo botle ba ngoana.

Contraindications

Maemong a mang, u ka se sebelisa lithethefatsi "Piracetam" (ente, liforomo tsa molomo)? sesebelisoa sena e sa o ile a bontša ka tabeng ea hypersensitivity (ho akarelletsa le derivatives tsa pyrrolidone), 'me lefu le Huntington e, ho hloleha renal, bokhachane, ferekanang ho tepella maikutlo, hemorrhagic leqeba , le ho nyantsha. Hape, lithethefatsi ena ha ea lokela ho fuoa bana ba ka tlaase selemo se le seng.

Mekhoa ea ho Sebelisa

Hona joale u tseba hore na ke hobane'ng "Piracetam" pilisi ka laetsoeng ho bakuli. Hona joale e lokela ho u bolella mabapi le kamoo sesebelisoa sa lokela ho nkoa ka.

Qalong ea phekolo piracetam tharollo ile laolwa entoe ka lethal dose ea la 10 g. Ka mor'a moo, ka tjhelete e ya moriana o lokolloa 'me ka isoa ka molomo. Hare ho ea amohela bolela pele ho ja ka litekanyetso li behoa ea mg, 800 (dihora tse 3). Ka mor'a ho ntlafatsa palo ea lithethefatsi e ne e fokotsehile ho 400 mg,. Ka nako ea phekolo ke libeke tse 6-8.

Re lokela ho hlokomela hore le litekanyetso li behoa ea letsatsi le letsatsi ea moriana o "Pyracetam" ka 'na ba e fapaneng' me ba itšetlehile ka mofuta le ho tiea tsa lefu lena. Mabapi le bolelele ba nako ea phekolo, ho feela rerang ngaka ho ea ka ho hlahloba ka ea meriana.

Ditshebeletso ho lokisetsa joalo laolwa sa feteng 30-50 mg, ka ho ya ka letsatsi. Tabeng ena, phekolo lokela ho nako e telele. Molomo tharollo fa ngoana makhetlo a 2 ka letsatsi (hoseng le mantsiboea). E lumelloa ho eketsa ya lero la tholoana kapa lino-mapholi tse ling.

liphetoho tse bohloko

E ka etsa hore tšebeliso undesired ea lithethefatsi "Piracetam"? Ente, hammoho le foromo molomo oa ea lithethefatsi ha e le hantle ba nang le bokhoni ba ho baka liphetoho boima. The hangata ho fetisisa o ile a bontša kenyeletsa tse latelang:

  • Metabolism: eketseha boima ba 'mele.
  • Makala kutloisiso e le tsamaiso ea methapo: otsela, hyperkinesia, ho tepella maikutlo, teneha kapele, mokhathala, pherekano, mabifi, ho robala meferefere, e ile ea eketseha ho kopanela liphate, ho tsekela, tremor, 'me hlooho e.
  • Tshilong ya dijo pampitšana: hlatsa, bohloko mpeng, letšollo le ho nyekoa ke pelo.
  • Letlalo: hypersensitivity.
  • Ajoa: hypotension, kgatelelo ya madi, gogoga ha pelo (a hlobaetsang le sethaleng).

overdose

Ha overdose "Piracetam" amplify liphello tsohle lehlakoreng. Ka kalafo sebelisa gastric lavage le ho noa ho bolela monya.

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