Bophelo, Litokisetso
Lithethefatsi 'Atenolol Nycomed'
Bakeng sa lithethefatsi "Atenolol Nycomed" ho na le lik'hemik'hale, 'me ho ea machaba selumisoa ka lebitso la "Atenolol". Ka puo ea litsebi tsa metsoako pharmacologists structurally lithethefatsi le hlaha e le (RS) -4- (2-hydroxy -3- (isopropylamino) phenyl-acetamide. Tablets "Atenolol" li emela oboevypuklye lipilisi tlotsitsoeng tsa 'mala o mosoeu, ba ka komiki sebopeho. The mele oa ka sehloohong ho fanoa hapa bakeng sa phomolo ea ka lehlakoreng le leng, ho na le matšoao AV55 le AV57.
Ka letlapa 'ngoe, ho itšetlehile ka mofuta o ho lokolloa ka ba le mashome a mahlano kapa lekholo milligrams ea atenolol. E le dikarolo ea thusang o ile a sebelisa talc, edible gelatin, propylene glycol, thaethaniamo dioxide, magnesium stearate, ipromeloza 2910 (15sP), poone starch, sodium lauryl sulfate, boima magnesium carbonate.
Medicine "Atenolol Nycomed 'liketso tse ka beta1-khetha (cardioselective) adrenoceptor thibela moemeli, lera botsitso mosebetsi hase. sesebelisoa sena se bontša antianginal, antiarrhythmic le hypotensive sebediswa. Ke khona ho thibela receptors beta-adrenergic pelo, fokotsa myocardial tlhotlheletso ya karohano le kutloelo-bohloko tsamaisong ea autonomic methapo le catecholamines, e potoloha maling. Medicine "Atenolol" phello fokotsa sinus automaticity, normalizes ea ho otla ha pelo ho eme e le nakong ea ho ikoetlisa. Sena stabilizes tshebetso le nyakallo ea contractility myocardial, slowing phello Av-conduction. Ka kopo lona ho na le ea fokotseha ka ya tlhokeho myocardial oksijene. Ka mokhoa o amohelehang ama hlophisitsoeng sebelisoa meriana "Atenolol" ka theola khatello ea mali. Tsitsisoa ha e le hantle antihypertensive le hlaha ho ea qetellong ea beke ea bobeli ea baeti ba fihlelang ho.
Ho lokisetsa "Atenolol Nycomed" holim'a mokhoa molomo baeti ba fihlelang ho ea nang le bokhoni ikakhele ka setotsoana pampitšana tshilong ya dijo ka bophahamo ba modumo ea 50-60% ea lethal dose tsamaisoa. Excreted ka moroto le halofo ea bophelo ba lihora tse la 6-7. linako tsena ka bakuli ba kholofalo renal, ho itšetlehile ka tekanyo ea karaoke set glomerular.
Bontšang bakeng sa lithethefatsi ke "Atenolol Nycomed" ke mefuta e meng ea kgatelelo ya madi le tachyarrhythmias (ho akarelletsa le sinus). Sebetsa meriana le ka moemeli e thibelang ho litlhaselo tsa angina.
The litekanyetso li behoa ea letsatsi le letsatsi ea lithethefatsi bakeng sa batho ba baholo ka ho phekola angina le kgatelelo ya madi fihla 50-100 mg,. matlapa a kenoa entse ho fihlela ho ka makhetlo a tse peli ka letsatsi ka lebaka la 'nete ea hore lethal dose ea letsatsi le letsatsi ba lokela ho sa feteng 200 mg,. Ho hlatsoa theoha lithethefatsi lokela ho ba e sa reng letho palo ya metsi.
moriana e sebediswa ho latela ka tieo le ka dikgothaletso tsa ngaka ho ba teng. Ba ikhopolang ho meriana e sa lumelloa. Lithethefatsi "Atenolol Nycomed" e na le litla-morao. Tsamaiso ea pelo le methapo ka arabela ponahalo ea meferefere bradycardia, Av-conduction, o ka ba le sensations tsa paresthesia le maoto le matsoho a batang, maemong a mang e bonahale matšoao a ha pelo. pampitšana tshilong ya dijo a leka ho hampe ho nyekeloa ke pelo ea lithethefatsi, pipitlelano, letšollo, e omeletseng molomo (seoelo), tsamaiso ea endocrine - ntshetsopeleng khoneha ya boemo ba motho ba hypoglycemic ka bakuli ba nang le lefu la tsoekere, urogenital oona tsamaisong - khoneha fokotseha ka potency. CNS bohloko liphetoho e ka bontša ho tšoaroa ke hlooho, molikoalikoane, ho mafu a robala, ho tepella maikutlo, maikutlo a ho ba le mokhathala. Hape, hoa khoneha ho mo kulisa, ho hlohlona, le redness. Maemong a kholiso mofufutso, phokotso e tabohileng secretion mokelikeli ile ha tlalehoa, ketsahalo e sa conjunctivitis.
Hape, ho na le a 'maloa a contraindications. Ka lethathamo bona kenyeletsa mekhahlelo motho ya ho hloleha foleng pelo, bradycardia, hypotension, li eketsehile ho nahanela ho lithethefatsi, 'me ba bang.
Boloka meriana sebakeng se ommeng, sireletswa ho leseli, se kenngwe ha bana. Kamoreng mocheso ho 25 ° C. lithethefatsi A lula thepa lona bakeng sa dilemo tse hlano.
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