BopheloLitokisetso

E atlehang antispasmodic "Papaverine Hydrochloride"

Ho lokisetsa "Papaverine hydrochloride" e bolela miotropnym ho bolela ho ba le matla spasmolytic sebediswa. Ka lilemo tse mashome a mangata, se sebelisoa ho fokotsa vascular molumo le mesifa boreleli boikhathollo le hoo e ka bang tsohle litho tse ka hare. E na le bitsoa joang bohato hypotensive. lithethefatsi ena dilates ea methapo, ho eketsa mali bophahamo ba modumo, haholo-holo bokong. lithethefatsi sena tekanyetso e phahameng ka tsela e hlollang ho fokotsa excitability a mesifa cardiac, hammoho le thusa hore ho slowing intracardiac conductivity. tšusumetso ea hae ka tsamaiso ea methapo e bohareng e bontša hanyenyane, le hoja ho na le phello e sedative ka tekanyetso e phahameng.

Lokolla ho lokisetsa "Papaverine hydrochloride" ka mefuta joalo litekanyetso li behoa:

- matlapa bakeng sa batho ba baholo 0,04g (10 likhomphutha.);

- matlapa Bana ba 0.01g (10 likhomphutha.);

- 2% ente (10 ampoules);

- rectal suppositories la 20 mg, (10 likhomphutha.).

Bontšang bakeng sa ho sebelisoa ke maemo a kang spasm ea litho boreleli mesifa peritoneum cholecystitis, renal colic; spastic colitis; endarteriite; bronchospasm; pilorospazme; vascular spasms, sebakeng bokong. Ka ho phekola angina pectoris bolela "Papaverine Hydrochloride" e sebediswa bakeng sa ho kopantswe phekolo le lithethefatsi tse ling.

Contraindications ho tšebeliso ea lithethefatsi ena ke:

hypersensitivity, phytoteratology sebete mosebetsi, glaucoma, bongoaneng (lilemo tse ho fihlela ho 0.5). Batho ba hōlileng ha baa lokela ho nka lithethefatsi ena ka lebaka la kotsi ya hyperthermia.

Le bolela "Papaverine hydrochloride": litaelo tsa tšebeliso

moriana o etsoang tsoa bakeng sa 3-4 leq. ka letsatsi. The litekanyetso li behoa bakeng sa tsamaiso ea se nang molekane oa matlapa a fapana le lilemo tsa mokuli. Batho ba baholo le beha matlapa lethal dose ea se nang molekane 40-60mg. Bana ba 0.5-2 g, - 5mg kela apotheek, 3-4 PM - 5-10mg, 5-6 k. -10mg, 7-9 a etsang dilitara tse. - 10-15mg, 10-14 a etsang dilitara tse. - 15-20mg.

Ente e laolwa intramuscularly kapa subcutaneously. Liente etsa 2-4 leq. ka letsatsi ke 1-2ml. Intravenous lithethefatsi tshelwa butle haholo ka 20mg pele phaella ka ho re tlhokeng sodium chloride 10-20ml (0,9% tharollo). Tsamaiso ena e molemo ka ho fetisisa etsoa tlas'a bookameli ba e le ngaka. Bakeng sa bakuli ba hōlileng ba se nang balekane lethal dose ea pele ba lokela ho sa feteng 10 mg,. Atisa ho ba ea lithethefatsi o laolwa parenterally hammoho le lithethefatsi tse fapa-fapaneng spazmaliticheskimi le analgesic, tse kang sethethefatsi "Promedol".

Likerese le papaverine laolwa rectally, 2-3 leq. 20-40mg ka letsatsi.

Ho lokisetsa "Papaverine hydrochloride" ho ka etsa hore liphello tse kang ho otsela, kulisa, arrythmia ventricular, upregulation tsa transaminases sebete, theola khatello ea mali, pipitlelano, eosinophilia.

Haeba matšoao a overdose hlokometse tse kang bofokoli kakaretso, diplopia, hypersomnia.

Ka ho sebelisa litaelo ena e khethehileng ho boloka lithethefatsi tseo khothalletsa tšebeliso hlokolosi lithethefatsi litsebeng bakuli le ba hōlileng; batho ba nang le likotsi hloohong, hypothyroidism, dysfunctions adrenal, a liphio le sebete; tachycardia; maemo a makala.

Lithethefatsi "Papaverine hydrochloride" nakong ea bokhachane 'me nakong fepa e molemo se ke a sebelisa ka lebaka la bohlokwa ba tsamaiso lona le polokeho linakong joalo e sa hlomamisoa.

Nakong ea phekolo, joala e thibetsoe. Ho tsuba nakong ea kalafo haholo ho fokotsa ho atleha ha moriana. Hammoho kenoa ho bolela "Papaverine" le "Dopegitom" ketso ea pele e haholo tsa fokotswa.

Papaverine hydrochloride e kenyelelitsoe a 'maloa ho kopantswe antispasmodics hammoho le lintho tse ling tse lithethefatsi:

- lithethefatsi "Lyupaverin" - le phenobarbital;

- lithethefatsi "Pafillin" - le platifillin gidrotata;

- ho lokisetsa "Kellatrin" - le kellinu le atropine sulfate ;

- lithethefatsi "Kelliverin" - le Kellin;

- ho lokisetsa "Nikoverin" - le asiti nicotinic.

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