Lithethefatsi "Metoprolol" litaelo bakeng sa ho sebelisoa e bua ka sehlopha se seng sa cardioselective beta-blockers hore na antiarrhythmic, antianginal le antihypertensive sebediswa. lithethefatsi Sena se nolofalletsa bakeng sa batlang e le khutšoanyane nako lieha ya Av conduction, fokotsa sinus noute automaticity, myocardial contractility le excitability le ho fokotsa lebelo leo pelo, khumo cardiac le myocardial oksijene. Ho phaella moo, cardioselective lithethefatsi "Metoprolol", theko ea tsona e ka bang leshome le metso e mehlano - mashome a mabeli li-ruble, ka katleho thibela le phello stimulatory tsa catecholamines ka pelo le khatello ea kelello-tlhaloganyo maikutlong le 'meleng. Ha e le ba ka sehloohong pharmacokinetic litšobotsi tsa lithethefatsi, mahloriso lona lebetsoeng le ka lero la mali e qala ho tla tšoauoa ka mor'a hoo e ka bang - lihora tse peli, 'me ho thoeng likarolelano halofo bophelo ho tloha lihora tse tharo ho isa ho tse supileng.
Hatisa hypotensive lithethefatsi "metoprolol" (taeo e pukwanana kamehla kenyelleditswe) ka mokgwa wa Pellets potoloha tšoeu-tranelate mmala le mofuta o mong oa tharollo ne a rerile hore morago ga moo e tsamaiso intravenous. Sebopeho sa lithethefatsi ena cardioselective e le motsoako o le mafolo-folo e kenyelelitsoe metoprolol tartrate. Tablets ho eketsehileng di na le dipegelo lactose monohydrate, microcrystalline selulose, povidone, k'halsiamo stearate, crospovidone le talc.
Sebelisa antianginal le antiarrhythmic "Metoprolol" litaelo bakeng sa ho sebelisoa e fanoeng ke moetsi o buella bakeng sa kalafo a bakuli ba tšoeroeng ke angina (ho akarelletsa le poso-infarction), kgatelelo ya madi le arrhythmias (ho akarelletsa mofuta supraventricular tachyarrhythmia). Ho phaella moo, hangata ha ho, lingaka ho laela le meriana hypotensive ho thibela litlhaselo tse migraine. Ea ho phekola e rarahaneng ea hyperthyroidism e boetse e khothalletsa hore ho qala ho fumana chelete cardioselective "Metoprolol". Ho bonahala reretsoe ho kenyeletsa bobeli tokiso phekolo mora infarction myocardial. Ena Melao ea kalafo ka e mong le e sebetsana le nyeoe motho ngaka beha feela ka motheong oa ditshekatsheko tsena.
Ha e le lethathamo la contraindications kholo ho ea hona joale cardioselective lithethefatsi tseo ke haholo-holo ho hlokahala hore ho abelwang karolo ya e nahanela eketsehile ho metoprolol tartrate, le alejiki itšoara joang ka metsoako leha e le efe ancillary. Batho ba nang le ho hloleha pelo, atrioventricular blockage, haholo sinus bradycardia kapa le literata sinoatrial ka tsela e tšoanang ha baa lokela ho nka e meriana antiarrhythmic "Metoprolol". Litaelo bakeng sa ho sebelisoa a boela sa kgothaletswa bakeng sa moemeli antihypertensive le sinus kula, maloetse a ya pheriferale ajoa mali tsamaisong kapa hypotension. Ba hlokolosi feteletseng lokela ho sebelisoa moriana ona tabeng ea hyperthyroidism, lefu la tsoekere mellitus, le asma e, pheochromocytoma, hypoglycemia, myasthenia gravis, emphysema, psoriasis, tshilong ya dijo acidosis, bao e seng alejiki la bronchitis kapa ho tepella maikutlo.