BopheloLitokisetso

Tablets 'Eufillin': bontšang bakeng sa tšebeliso

"Eufillin" Tablets ke Adenozinergicheskie ho bolela, 'me synonymes bona ke "Aminophylline, Escom," "Aminofilliin" "Euffillin-Darnitsya". Ba ka sehloohong a sebetsang a ntho lokisetsa ka holimo o sebeletsa aminophylline le tlaasana - acid e stearic le starch litapole.

"Eufillin": tlhaloso ya moriana

lithethefatsi ena e na le phello mesebetsi e sa tšoaneng 'meleng. Eufillin di hlohleletsago sa tsamaiso ea methapo e bohareng, eketsa contractile myocardium mosebetsi, o khanna katoloso ea renal, gogoga le pheriferale methapo ea mali, thusa ho khatello ka mothapo ho methapo theola, 'me e haholo ho eketsa renal phallo ea mali. Hape, "Eufillin" matlapa a ba le e leka-lekaneng diuretic e le hantle, thibela metsoako platelet aggregation, thibela metsoako lokolloa ha palo seleng ea instigators allergy. Ho decreases le contractile mosebetsi oa mesifa le boreleli, 'me kahoo ho phomola le bronchial methapo le ho tlosa bronchospasm. O ile a re ho lokisetsa e hantle ananelang, 'me mahloriso lona lebetsoeng le maling le hlaha ka hare ho lihora tse peli ka mor'a hore tsamaiso ea, empa leha ho le joalo, e boetse e ho itima lijo metabolised ke sebete, moo metabolites khathetseng moeeng ba thehoa. About 10% ea lithethefatsi o ile a fumana e excreted sa fetohe ka moroto wa.

Tablets "Eufillin": ba bonahala

sehlahisoa sena e reretsoe ho sebelisoa ka ho ba teng ha bronchospasm le asma e, le asma e cardiac, kgatelelo ya madi etsahalang ka ajoa methapo, haeba litlhaselo tsa tsamaya bronchospasm le mafu a matšoafo tsa Cheyne-Stokes. Ba ile ba boela li sebelisoa tabeng ea hlokahala hore ba ho ntlafatsa ajoa ka likopi bokong 'me bakeng sa ho imoloha tsa maqakabetsi bokong vascular, ba fokotsa khatello intracranial, edema bokong, e leng hlaha ka leqeba ischemic kapa ha ho hlōleha foleng oa phepelo ea mali bokong.

"Eufillin" pilisi: litaelo bakeng sa tshebediso ya moriana

Lithethefatsi e nkiloeng ka molomo, hang feela ka mor'a lijo, makhetlo a isa ho a mararo ka letsatsi, le lethal dose bakeng sa batho ba baholo ke dikgerama 0,15. The lethal dose ea se nang molekane bakeng sa mamello batho ba baholo ba ka 'na sa feteng 0.5 g, Children amohetse ho lokisetsa lethal dose fokotswa ho 7-10mg / lik'hilograma le tshwerweng bakeng sa tekanyetso 4 motšehare. Bakeng sa bana ka mohato o le mong lethal dose le 'ngoe e ke ke e phahameng ho feta 7 mg, / lik'hilograma.

Ha ho hloka mosebetsi ea litsamaiso biotransformation potlakisang tsebetso ea lik'hemik'hale ea sebete ka bakuli ba fetang lilemo tse 55 ba lilemong tsa ho le neonates, lithethefatsi "Eufillin" abeloa ka hloko haholo.

Le litla-morao, e leng ho etsa hore matlapa ao "Eufillin"

Ha o dumella ho baeti ba fihlelang ho ea le moemeli ka mpeng letho, ho ka hlaha le matšoao dyspeptic, tse amanang le halefisa lithethefatsi thepa. Hape tabeng ea nahanela phahameng ho ethylenediamine ka 'na la hlaha dermis exfoliative kapa febrile itšoara joang.

Contraindications

Ho sebelisoa ha lithethefatsi ena e contraindicated ka lefu la sethoathoa, hypotension matla, arrhythmia le tachycardia paroxysmal. U se ke ua nka matlapa "Eufillin" ka ho ba teng ha ho hloleha pelo, haholo-holo haeba e amana le infarction myocardial, hammoho le ha ho na le pelo morethetho boloetse, kapa gogoga insufficiency.

Overdose "Eufillin"

Ka ketsahalo ea overdose ho na le matšoao a kang letšollo, bohloko epigastric, ho ipolaisa tlala, mali gastrointestinal, ho nyekoa ke pelo, restlessness, tachycardia, generalized tsitsipana, arrhythmia ventricular, e phallang ea sefahleho, ho hlatsa, lefu la ho hlobaela, hipnoe le photophobia.

Maemong ana, o lokela ho hang-hang khaotsa tshebediso ya lithethefatsi "Eufillin" 'me ba qala ho susumelletsa excretion lona le' mele, e leng ke ho hlokahala hore ho hlatsoa tsoa ka mpa, le tšoare ka e qobelloang diuresis, hemosorption, plasmasorption, hemodialysis, peritoneal dialysis, le kalafo ebe bontshang matshwao.

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