BopheloLitokisetso

"Mydocalm": hore na o thusa, tlhaloso ea moriana, contraindications

ke lithethefatsi "Mydocalm" ke efe? Ka sona se etsang hore sesebelisoa see? Ho bonahala le litšobotsi tsa lithethefatsi ena, re hlahisa mona ka tlase. U tla boela u ithute ka mokhoa oa ho alafa lithethefatsi sena, kamoo ho fana le seo e se fupereng.

Foromo ya lithethefatsi lokolloa, ambalaji, tlhaloso, sebopeho

Ka mofuta ofe ho famasi lithethefatsi "Mydocalm" fihla (ho tloha ho se thusa moriana ona, re ka hlalosa mona ka tlase)? sesebelisoa ke fumaneha ka matlapa a le hape ka tharollo e ne a rerile hore tsamaiso parenteral.

Round le tšoeu "Mydocalm" letlapa, theko ea eona e bontšitsoeng tlaase mona, e na le tolperisone hydrochloride. Ka metsoako 'ngoe ea moriana li nkoa: anhydrous colloidal silicone, acid e citric monohydrate, starch poone, stearin, hydroxypropylmethyl selulose 2910, talc, Macrogol 6000, microcrystalline selulose, colorant, lactose monohydrate le thaethaniamo dioxide.

Fumaneha ka dipakete blister ke mokhoa, tse kenngoa ka mabokose a entsoe ka pampiri.

The tharollo e hlakileng "Mydocalm" ka ampoules boetse e na le tolperisone hydrochloride le lidocaine. Ho phaella moo, lithethefatsi kenyeletsang metsoako latelang: talc, acid e citric monohydrate, lactose monohydrate, silicone colloidal anhydrous, macrogol 6000, microcrystalline selulose, stearin, thaethaniamo dioxide, starch poone, oxide e ba batsho tšepe, hydroxypropylmethyl selulose 2910, tšepe oxide e le lefubedu le le bosehla tšepe oxide e.

Lithethefatsi "Mydocalm" ka ampoules tse lik'hontheinara polasetiki, tseo ba kenngoa ka mabokose a entsoe ka lebokoso.

thepa senotlolo

le "Mydocalm" ke eng? Ka etsa hore lithethefatsi ee? Ho ea ka litaelo tseo, ka taba moemeli bolela relaxants mesifa aminoketonovoy sehlopha eo e na le phello e bohareng.

The bohlokwa ba tsamaiso ea lithethefatsi ena e amahanngoa le molao oa tsamaiso ea mosebetsi oa karolo e itseng (caudal) ya sebopeho reticular. Tshebediso ya moriana o ka khothalletsa batho thibelo ea eketseha excitability tsa reflex lesapo la mokokotlo. E boetse e ama methapo ea kutlo (pheriferale).

Features lithethefatsi

Ho lokisetsa "Mydocalm" (sebeletsana oa sesebelisoa le tse ling tse amohelehang, empa tlas'a maemo a itseng) e H-anticholinergic. moemeli lona a sebetsang a na le phello e tiileng ka lera ea likhoele mathomo (afferent), le motoneurons. e le hantle sena ke ka lebaka la lithethefatsi ke matla a ho susumetsa mosebetsing oa reflex synapses lesapo la mokokotlo.

Hape ela hloko hore lithethefatsi hona ka lekhetlo la bobeli liehisa neurotransmitters. Hlahellang ka lebaka la ho thibelo ya khalsiamo thulaganyou e kena ka sebopeho synaptic, tse teng ka likhoele methapo ea kutlo.

Phello ea lithethefatsi tseleng reticulospinal ke haholo-holo ho phatlalatsoa ha decelerating dithulaganyo nyakallo. Ka tsela e tšoanang mestnoanesteziryuschee lemoha le ho etsa lintho tsa moriana (ka lebaka la ho dikahare tsa lidocaine ho eona).

The kinetics ya moriana

moemeli li nkoa e le e hantle ananelang tloha eyeglobe ena. mahloriso lona (, max) e ile ea fihla ka mor'a metsotso e 65 ka mor'a ho nka mali. metabolism lithethefatsi le hlaha ka sebete 'me liphio. Tolperisone derivatives hlaha ka moroto wa.

Pheta nete hore "Mydocalm" ha e na phello liphio le sebete, hammoho le tshebetso ya ho hematopoiesis.

sesebelisoa sa decreases ho se tenyetsehe le ho experimentally hlohlelletsoa mesifa hypertonicity. Moriana thepa ea lithethefatsi li sebelisoa haholo ho fokotsa mesifa tsitsipano le pathological hypertonus hore li amahanngoa le mafu a extrapyramidal.

Ho lokela ho hlokomeloe hore lithethefatsi kgothaletsa mosebetsi oa motho (mekhatlo hae). Ho phaella moo, bo se na le phello e cortex bokong, ka botlalo ea bolokelang ba boemo ba falimehe ba mokuli.

Ho latela thuto, kalafo "Mydocalm" hlahisa hanyenyane bitsoa antispasmodic le adrenoceptor thibela liphello. Ka lebaka la sena, ho ba ntlafala dinama tse nyenyane tse perfusion.

Ha ba ntse ba thulana le liteko tse nako e telele ea tleleniki ea moemeli ena ne ba se na le tšusumetso e bitsoa ka mali le liphio.

Lithethefatsi "Mydocalm": seo thusa?

sesebelisoa e bontšitsoeng bakeng sa ho sebelisoa maemong a latelang:

  • Ikatisetsa kokelo ea bana, ka sepheo sa ho lefu phekolo Little o (khr, spastic shoele litho). Ho phaella moo, lithethefatsi ena e sebelisoa ka fapaneng hlahang ho yona magazine le matšoao a dystonias mesifa.
  • Tlas'a maemo a hore ba tsamaea le hypertonus pathological tsa striated mesifa dinama tse nyenyane tse e loketseng ho pathologies tsoelang pele (methapo ea kutlo) manyolo (mohlala, ke multiple sclerosis, encephalomyelitis, myelopathy, barrel liphello tsa setorouku, pyramidal pampitšana diso).
  • Tlas'a maemo a eo ba ipotsa ka lebaka la ho senya vascular innervation (mohlala, acrocyanosis, angioneurotic disbazii hill tlhaho).
  • Ha mesifa hypertonicity, contracture mesifa eo felehetsa mafu a litho tsa ka hare ho tsamaea (mohlala, spondylosis, ramatiki ba litsoeng, lengole le manonyello a liqholo, spondylarthritis, syndromes tsa lumbar le cervical).
  • Ha poso-thrombotic venous phallo ea mali mafu a le lymphodynamics.
  • E le ho fokotsa postoperative kalafo ka masapo le ho sithabela ho itlhakisa.
  • Ha liso trophic thehoa ka lipheletsong tse tlaase, ke angiopathy (ho akarelletsa le diabetogenic), thromboangiitis obliterans angiosclerosis le, hammoho le mafu autoimmune (lefu Raynaud le systemic sclerosis).

Ho thibeloa tšebeliso ea

Maemong a mang, u sitoa ho abela le pilisi, injectables "Mydocalm"? Ho sebelisoa ha lithethefatsi ena e contraindicated ka se:

  • myasthenia gravis;
  • hypersensitivity ho tolperisone le kulisoa tsebisoe lidocaine;
  • tlaase ho lilemo tse likhoeli tse tharo (foromo Letlapa ho selemo se le seng).

Dosing

Sekemeng oa sesebelisoa e beha ngaka ho itšetlehile ka le lefu lena, 'me tolerability lithethefatsi.

Bakeng sa batho ba baholo moriana o laolwa ka palo ea 150-450 mg, (letsatsi le letsatsi lethal dose) ka mehato e meraro. The litekanyetso li behoa qalang tsa meriana ena ke 50 mg, ka makhetlo a mararo ka letsatsi. Ka lebaka la ho hloka e sebetsa le keketseho ea lona.

Bakeng sa ente intramuscular, lithethefatsi e sebediswa ka palo ya mg, 200 ka letsatsi (tse peli ente) le intravenous - 100 mg, (hang ka letsatsi). Tabeng ea bobeli e hloka Infusion lieha haholo ya moriana.

Bakeng sa bana ba baholoanyane ho feta likhoeli tse tharo (ho fihlela ho lilemo tse 6) le litekanyetso li behoa ea ea lithethefatsi le tlas'a ho nahanela e balwa ka tsela e latelang: 5,10 mg, ka ho ya ka lik'hilograma boima ba 'mele (ka makhetlo a mararo letsatsi le letsatsi). Ngoana lilemo tse 7-14 buelloa ho sebelisa letlapa ka lethal dose ea letsatsi le letsatsi ea 2-4 mg, ka ho ya ka lik'hilograma tsa 'mele (ka makhetlo a mararo letsatsi le letsatsi).

tsamaiso molomo "Mydocalm" le lokela ho ho kopantswe le lijo.

lehlakoreng bohato

Etellang lithethefatsi le hypersensitivity motho a ka bakela bofokoli ka mesifa, liketsahalo dyspeptic ea tlhaho (ho nyekoa ke pelo, boemong bo sa thabiseng le ho hlatsa) le hlooho.

Ka potlako intravenous tharollo Infusion ka 'na fokotseha khatello ea mali.

Haeba u hypersensitive ho moriana hlahisa kulisa. E le busa, tekanyetso e nyenyane ea litla meriana lehlakoreng ke ho itima lijo haholo.

ditshebeditsano lithethefatsi

Tlhahisoleseding e mabapi le sebelisana, e leng lekanyetsang tshebediso ya sehlahiswa sena ke ha e fumanehe. Leha ho le joalo, re lokela ho hlokomela hore tolperisone e susumetsoa ke tsamaiso ea methapo e bohareng. Kahoo lithethefatsi hase eena ea bakang ho otsela, kahoo, ho ka kopanngoa le hypnotic le sedative, hammoho le medicaments nang ethanol e.

Ha tsoa hong tsamaiso "Mydocalm" acid e niflumic kgothaletsa phello. Haeba ho hlokahala, e le motsoako oa mahlahana a joalo a ka hlokang phokotso lethal dose ea bobeli.

Pheriferale mesifa relaxants, lithethefatsi bakeng sa thethebatso kakaretso le dintho psychotropic, hammoho le "clonidine" ntlafatsa ho atleha ha tolperisone.

Theko le ulasan pelanggan

Ke bokae "Mydocalm"? Theko ea moemeli ena ke ka 185 li-ruble.

Testimonials stipulate hore lithethefatsi potso bontša ka boeona e ka tsela e atlehang haholo, haholo-holo ka mafu a manonyeletso. Ho phaella moo, ke sesebelisoa sena se molemo haholo bakeng sa ho ajoa mali bokong, ho akarelletsa le itlhahela ka mor'a ho lemala boko sithabetsang.

Har'a ulasan pelanggan mpe ka ho tsejoa ke batho hore re lithethefatsi "Mydocalm" hase panacea. Hangata ka ho fetisisa, meriana ena e sebelisoa e le kalafo ya tlhokomelo.

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