BopheloLitokisetso

Fenkarol. Litaelo tsa tšebeliso

Fenkarol taeo e pukwanana amana derivatives hinuklidilkarbinola. O ne a nka moriana o, ho fapana le maemo a antihistamines, activates diaminoksidazu - potlakisang tsebetso ea lik'hemik'hale cleavable tridtsatiprotsentnogo dinama tse nyenyane tse ho histamine.

Sena se ka hlalosa phahameng phekolo phello ea ho moemeli maemong moo lithethefatsi tse ling tse u se ke ua felisa bothata. E boetse e ile a bolela hore ka nako ea ho pepesehela bona ho lithethefatsi ena o phahametse meriana "Diphenhydramine".

Fenkarol (mosebedisi ya kopo ya e na le boitsebiso bo mabapi le ena) ho fokotsa mosebetsi likokoana-hloko tsa histamine. mokhoa fokolisa matla a ho spasm ea mesifa boreleli ka e ntse likahare ka 'me tsa fokodisa le e lumellang metsi ho kena ea methapong. O ne a nka lithethefatsi o holinoliticheskoe protivoserotoninovoe le phello 'mele,' me hape felisa ho hlohlona le desensitizes.

Fenkarol (litaelo bakeng sa ho sebelisoa e haholo-holo o ile a hlokomela) ha e ama ho sebetsa ha tsela nyahamisa ho tsamaiso ea methapo e bohareng le e ka boko ba ka sebelisoa ho fumana lintho tse ngata fokolang haholo - ka tlase ho ya 0.05%.

The moemeli thuto.bafuputsi ba meriana e na le matla a ho potlako ikakhele ka setotsoana pampitšana tshilong ya dijo (bonyane 45%). Halofo ea hora lithethefatsi lemoha ka lisele tsa 'mele. Ho 'nile ha e thehilweng hore e moholo serum dikahare fihla ka mor'a metsotso e mashome a mane a metso e mehlano ka mor'a dosing.

Fenkarol (taeo e pukwanana bontša ena) concentrated haholo-holo ka ea matšoafo, sebete le liphio. The dikahare nyenyane ka ho fetisisa lithethefatsi bokong.

moriana o metabolized ka thepa sebete. Fetisisa excreted ka bile, moroto, 'me ke methapo ka hare ho lihora tse mashome a mane a metso e robeli ka mor'a a e-ja (liphesente tse mashome a mane a metso e mene ba moemeli molemo). Le mantle tsoa karolo eo ea lithethefatsi, e leng ha e so adsorbed.

The moemeli a thuto.bafuputsi meriana bontša bakeng sa ho sebelisoa e le lijo le lithethefatsi mefuta kulisoa, feberu furu, hives (bobeli a hlobaetsang le a sa foleng), angioedema, feberu furu, alejiki rinopatii, dermatosis, eczema, psoriasis, atopic dermatitis, liso tsa ka maleng letlalo, maloetse a tšoaetsanoang-alejiki holimo mathata a ho hema bronchospastic motsoako.

moriana kgothaletswa bakeng sa ho sebelisoa ka ho toba ka hare postprandial. Fenkarol bakeng sa bana (pukwanana bontša ena) bontša milligrams hlano hang ka letsatsi, empa haeba mokuli a lilemo - ho tloha selemo se le seng ho lilemo tse tharo, ka palo palo yohle ha ho feta milligrams lesometlhano. bakuli Young tloha tharo ho isa ho tse supileng - milligrams leshome ka makhetlo a mabeli ka letsatsi, ho tloha a supileng ho leshome le metso e - tse leshome ho lesometlhano milligrams ka tekanyetso e meraro (letsatsi le letsatsi lethal dose - ha ho feta mashome a mahlano, mg), tse fetang leshome le metso e - mashome a mabeli kapa tse mashome a mabeli a metso e mehlano milligrams hang ka letsatsi (empa e se mg, tse fetang lekholo).

Ka nako ea 'nete hore phekolo hangata ho tloha matsatsi a leshome ho leshome le metso e mehlano. Ha eba ho kalafo hlokahala o etsoa ka makhetlo-khetlo.

Tabeng ea inadvertent tlolela ba amohelang molaetsa tlang ho bolela o tsoela pele ho sebelisa moriana o ka ntle e ntseng e eketseha lethal dose.

Lithethefatsi "Fenkarol" nakong ea bokhachane e contraindicated. Hape, ho e sa ba laela hore hypersensitivity mokuli a se ho entsoe.

litla khoneha lehlakoreng. Ba bontša ka setotsoana ho mucosa tsa molomo omile, dyspepsia, tse tlosoa ka mor'a emisa tshebediso ya moriana. E a hlokomela hore monyetla oa liphello tse bohloko ke phahame ka ho batho ba nang le mafu a ea tsamaiso tshilong ya dijo.

O ile a re moemeli meriana ha e ntlafatsa phello ea joala le lithethefatsi hypnotic. Ho ntlafatsa absorption ea lithethefatsi le tse tšoauoa ka ea liehang hapang.

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