Bophelo, Litokisetso
"DITT depo": litaelo bakeng sa ho sebelisoa, contraindications, litla-morao, recensioni, lifoto
Ke eng seo u se tsebang ka meriana ena, tse kang "DITT depo"? Litaelo tsa tšebeliso, contraindications, ulasan pelanggan le ditlamorao tsa ea lithethefatsi ho tla buisanoa ka ho eketsehileng.
Ambalaji le mofuta o mong oa lithethefatsi e, sebopeho lona
Ka seo foromo lihlahisoa sethethefatsi ka "DITT depo"? Litaelo tsa litlaleho tse sebelisoa e ka rekoa ka mokgwa wa e tharollo mafura bakeng sa ente intramuscular. Ba ka sehloohong a sebetsang a motsoako oa lithethefatsi ena ke fluphenazine decanoate. Ha e ntse e kena ka rekisa ampoules lefifi khalase, pele ho tsa phutheloa ka seleng ea moeli le pampiri dipakete, ka ho latellana.
pharmacology
ke thepa le moriana tlholeho moriana o "DITT depo" ke efe? Litaelo tsa tšebeliso, ulasan pelanggan re ena ke nako e telele-ho nka bohato meriana antipsychotic. Ho ke oa sehlopha sa batho ba neuroleptics polyvalent le lipontsuoa bitsoa antipsychotic thepa, tse ho kopantswe le thunye le phello antiemetic. Hape, lithethefatsi ena e na le e le bonolo le phello sedative.
Ke'ng se etsang hore ho atleha ha lithethefatsi "DITT depo"? Litaelo bakeng sa ho sebelisoa e bolela hore liphello tsa eona antipsychotic amanang le thibela likepe tsa dopamine D2 receptors Mesocortical le litsamaiso mesolimbic.
Sedative thepa ea lithethefatsi ena ba bolela hore ka tekano le feela o ile a re ha tekanyetso e phahameng ea tharollo. Ba ka lebaka la ho se thibela likepe tsa receptors adrenergic dikarolo tsa motho ya bakoang boko.
Mabapi le liphello tse-ba khahlanong le emetic tsa meriana, joale e e amahanngoa le ho se thibela likepe tsa dopamine D2 receptor thunye libaka tsa setsi sa ho hlatsa. Ho lokela ho hlokomeloe hore phello hypothermic ea lithethefatsi ena e bontša se thibela likepe tsa dopamine receptors tsa hypothalamus le.
Bakae lithethefatsi e qala ho etsa lintho "DITT depo"? Litaelo tsa (tharollo Foto ente fanoa ka pampiri ena) tšebeliso o tlaleha hore e le hantle phekolo ea lithethefatsi e hangata ile a bontša ka mor'a lihora tse 25-72 ka mor'a ente e. Ho lokela ho hlokomeloe hore ho thepa ya lithethefatsi antipsychotic tlas'a ho nahanela ba ho fetisisa le bitsoa joang ka nako ho tloha lihora tse 49 ho ea 97 ka mor'a tsamaiso ea tharollo.
The kinetics ya moriana
bath ya pharmacokinetics ea lithethefatsi "DITT depo" ke eng? Litaelo bakeng sa ho sebelisoa tsa batho ba reng bo fluphenazine ka mokgwa wa e phahameng ea limolek'hule boima Ester oli tharollo ea mafura acid e ka kgona ho ipokellela ka adipose didepo, hammoho le butle lokolloa botlamuoeng.
Mora entoe nameng ya ea mahloriso palo e kahodimodimo ea elements e fihlellwa ka mor'a lihora tse 25 ka lero la mali. Tabeng ena, fluphenazine tlama ho phepelo ea mali ka ho 90%.
O ne a nka lithethefatsi habonolo lifapano le mokoallo placental le fetisa ka mali-boko, 'me ha ba excreted ke hemodialysis.
Fluphenazine ho feletseng 'me haholo metabolised ke tsamaiso ea sebete potlakisang tsebetso ea lik'hemik'hale e amang cytochrome P450. Le 'mele e excreted le bile le moroto. metabolites mafolofolo elements ena e sa utloisise ka ho feletseng.
Fluphenazine halofo bophelo bo lihora 7-10.
ya litatoli na
Maemong a mang, ho ba le mamello e hlophisitsweng liente "DITT depo"? Litaelo bakeng sa ho sebelisoa e bolela bopaki bo kang:
- exacerbation ea bokuli ba ho kopana hlooho (bakeng sa thibelo ya);
- ka nako e telele ya tlhokomelo kalafo ea bokuli ba ho kopana hlooho foleng.
Ho thibeloa tshebediso ya
meriana talingoa e thibetsoe maemong a latelang:
- tlas'a mafu boima SS, ho akarelletsa le decompensated foleng ho hloleha ho potoloha ha mali 'me hypotension;
- a sa le nahanela phahameng tsa mokuli hore fluphenazine le, hammoho le ho likarolo tse ling tsa moriana;
- hateletsoeng nakong ea CNS le re comatose;
- nakong ea bokhachane;
- ka ho sithabela lehata le bo tsoelang pele e le mafu systemic tsa boko le lesapong la mokokotlo;
- ka ho iphepa;
- le litsebeng sebete mosebetsi le tsamaiso ea mali;
- ho fihlela ho lilemo tse 12.
Hloko ho sebelisa lithethefatsi
Ba qoaile "DITT depo 'lithethefatsi tseo ke li behetsoeng:
- bokhoba ba tahi, hammoho le eketseha susceptibility ho liphetoho hepatotoxic;
- liphetoho pathological maling, hammoho le ka tlōla hematopoiesis;
- kulisoa phenothiazines, ho akarelletsa histori ea;
- koalo glaucoma;
- kankere ea matsoele;
- e amanang le sebete le / kapa ho hloleha renal;
- liso tsa ka maleng tsa pampitšana tshilong ya dijo, ho akarelletsa le nako ea ho kula a hlobaetsang;
- prostatic hyperplasia le liponahatso tsa tleleniki;
- myxedema;
- maloetse, a tsamaea le mathata thromboembolic;
- lefu Parkinson;
- boloetse bo sa foleng ka ho hema ho hloleha (ho akarelletsa le bana);
- lefu Reye ya;
- sethoathoa, ho hlatsa, sethoathoa;
- cachexia;
- ka botsofali.
The tharollo ea lithethefatsi "DITT depo": litaelo tsa tšebeliso
The ampoules ea lithethefatsi ena e reretsoe ho dithuto tsa nako e telele tsa phekolo (bonyane likhoeli tse tharo). lethal dose ea hae ka lekhetlo la pele ho bakuli ka ho fetisisa ke 12.5-25 mg,. Morago ga moo e tekanyetso, hammoho e le karohano pakeng tsa liente ea tharollo ikemiselitse itšetlehileng ka phello phekolo.
Kalafo ea bakuli le hypersensitivity ho phenothiazines lokela ho qala ka masene haholo.
Ea seng a hōlile e hloka ho kgethwa ha tekanyetso tlaase ho feta bakuli ba ka tlaase (hoo e ka bang 1/4 ho 1/3 ya dosing le). Tabeng ena ka mor'a tsona hloka tlhokomelo ka linako tsohle.
Liketsahalo ka tlhaku
The tharollo ea lithethefatsi "DITT depo" ho ka etsa hore tse latelang tse sa rateheng itšoara joang:
- extrapyramidal lefu, akathisia, tardive dyskinesia, dystopia, maqakabetsi oculogyric, hyperreflexia, opisthotonos;
- neuroleptic bolaeang lefu, e leng e ka ba e bolaeang;
- orthostatic hypotension, ho fufuleloa, liphetoho khatello ea mali, ho nyekoa ke pelo, hypotension, tahlehelo ea takatso ea lijo, glaucoma, salivation ka tsela e feteletseng, atony senya, polyuria, mantle a obstruction, molomo o omileng, tachycardia, hlooho e opang, pono thothofatsang, pipitlelano, nasal tsubuhlellano;
- arrhythmias ventricular, ka tšohanyetso lefu, ventricular tachycardia, cardiac tšoaroe;
- e sa tloaelehang diabolololo, pheriferale edema, lefu la matsatsing, hyponatremia, ho hloka matla tseo e leng banna, liphetoho tse ka boima ba 'mele, liphetoho libido ka basali;
- pruritus, exfoliative dermatitis, etymology, seborea, urticaria, anaphylactic liphetoho, photosensitivity, angioedema, bronchial spasm, laryngeal edema;
- agranulocytosis, leukopenia, cholestatic nyooko;
- sethoathoa, feberu, liphetoho ECG, etsolloa diskinenziyu, ho hlatsa, venous thromboembolism, lupus-joaloka lefu, 'me ba bang.
Testimonials
Hona joale, u lokela ho tseba, ho tloha etse'ng Shots "DITT depo." Litaelo tsa tšebeliso, litla-morao, 'me contraindications ho tshebediso ya tharollo ena e boetse e tšohla ka holimo.
Ho ea ka bakuli ba neng tšoaroa ka lithethefatsi tse sa tšoaneng antipsychotic, lithethefatsi "DITT depo" o sebetsang haholo ka tsela e atlehileng haholoanyane le ho tlosa matšoao mpe kaofela bokuli ba ho kopana hlooho. Ho qaloa ho lithethefatsi ena o tsitsitse haholo 'me ka nako e telele ho leballa motho.
The drawback feela oa sesebelisoa sena ke o moholo o ka tlhaku liphetoho. Ka matsatsing a pele a oa phekolo ka ho batho ba bang ba tšoaea hyperthermia, kgatelelo ya madi le autonomic ho se sebetse. Hape, bakuli ba bangata ba bone ho mesifa giperkinezy tsa molomo le sefahleho, smacked molomo oa hae le leleme sisinyehang. Ho feta moo, ho sebelisa lithethefatsi ena e atisa ho ile a etsa hore ho tepella maikutlo ea sa tšoaneng ho tiea.
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