Bophelo, Litokisetso
"Artrokol" (gel): litaelo bakeng sa ho sebelisoa, analogs le ulasan pelanggan
Ke lokela ho sebelisa lithethefatsi "Artrokol" (gel)? Litaelo bakeng sa ho sebelisoa tsa lithethefatsi li tla hlalosoa ka sehlooho sena. Hape, u tla ithuta ho se ileng sa meriana e beuweng bakuli, hore na o na le analogues le maikutlo leha e le efe mabapi le ho siea mosebedisi.
Formulations, lithethefatsi diphuthelwana le sebopeho lona
"Artrokol '- gel (2,5%) bakeng sa ho sebelisoa ka ntle. Ka ho rekisa e fihla ka aluminium tube, 45 e ne e le teng le ho lebokose lebokoso hammoho moriana ke pampitsana le litaelo tse hlakileng ho sebelisoa.
Hore na e Link lithethefatsi "Artrokol" (gel)? 100 g, ea mahareng ena e ne e ena 2,5 g, ea motsoako o sebetsang, e le ketoprofen. Ho phaella moo, ka lithethefatsi ka eona ho kenyeletsa tse latelang tšehetso likarolo: trolamine, Carbomer 980, 96% ethanol, metsi a hloekisitsoeng le methylene parahydroxybenzoate.
Molao-motheo oa tšebetso ea moriana o ka
"Artrokol" - e gel, ea motsoako o le mafolo-folo e ketoprofen. Itse moriana o ho matleng a sehlopha sa lithethefatsi nonsteroidal-ba khahlanong le a hlabang, hammoho le derivatives ea acid e arylpropionic.
Base lintho tse bonahalang ho nkoa moriana o fana ka-ba khahlanong le a hlabang le analgesic le hantle, eo e hlaha nakong ea thibelo bao e seng khetha ya Cox-1, bradykinin le Cox-2, le lera tsitsisoa (lysosomal) le thibelo ya macrophage falla.
Ho phaella moo, lithethefatsi "Artrokol" (gel) hlahisa thepa-ba khahlanong le a hlabang le moriana o thethefatsang kutlo. Ho kgona ho ho sebetsa ka hoseng 'me a morao seleng ea vascular mohato ea ho a hlabang. Hape, lithethefatsi ena liehisa platelet aggregation.
Litšobotsi pharmacokinetic ya
Ho latela litaelo le khomaretse, ketoprofen (ba mafolofolo motsoako oa moriana o le) ka mora kopo ea lihlooho tsa puisano ho letlalo e ananelang, 'me joale le kenella ka hare ka e le setsi sa tsamaiso e hlabang le nakong ea nako e telele lula le lakatsa mahloriso phekola ka lisele tse ka.
Absorption ya lithethefatsi ka ajoa systemic e fokolang haholo (ka 5% ea lethal dose ka sebediswa). Tabeng ena, ho absorption ka kemisong ea mali o lieha haholo.
Ea mahloriso ba mafolofolo motsoako oa moriana (ho sebedisa 50-150 mg, ea ketoprofen) maling ka mor'a lihora tse 7,5 ke 0.08-0.15 feela mg, / ml tse.
Lithethefatsi "Artrokol" (gel) le morero oa oona?
The bontšang bakeng sa tshebediso ya gel tlas'a ho nahanela ba e bolela tse latelang:
- myalgia, rheumatic le rheumatic hlahang ho yona;
- mafu a ea tsamaiso ea musculoskeletal (ho akarelletsa e ruruhisang ramatiki, articular syndrome, nakong exacerbation gout, ankylosing spondylitis, psoriatic ramatiki, osteochondrosis, tabanan ya selegae le fapaneng, a hlabang lethopa tsa tendons, ligaments, sciatica, bursitis kapa lumbago);
- karolo ea kalafo e rarahaneng ea hlabang pathologies methapong (mohlala, phlebitis, periphlebitis), lisele tsa mmele nodes kapa lijana lisele tsa mmele (mohlala, lymphangitis, ka ntle feela lymphadenitis);
- poso-sithabetsang ho ruruha ea tsamaiso ea musculoskeletal le dinama tse nyenyane tse bonolo (ho akarelletsa le kalafo bontshang matshwao ya dikotsi bonolo, ho akarelletsa le sprains, likotsi lipapali, sprains kapa meokho ea tendons le ligaments, matetetso, poso-sithabetsang bohloko).
Ho thibeloa tshebediso ya
Seo ha "Artrokol" mafura thusa, re o ile a hlalosa ka holimo. Leha ho le joalo, sena se bolela ho na le contraindications. Tsena li akarelletsa tse latelang:
- lilemo tlas'a lilemo tse 12;
- phahameng nahanela ho thepa ea motheo ea lithethefatsi hammoho le asiti acetylsalicylic le NSAIDs tse ling;
- le trimester karolo ea boraro ea ho ima le kanyeso.
Lithethefatsi "Artrokol" (gel): litaelo tsa tšebeliso
Bakeng sa kalafo ya gel e hlobolisa 5.4 cm, nako e telele ka eona ho bolela ho etsa kōpo ea ho ea letlalo ka sebaka lakatsa le bonolo hohla massaging mekhatlo fihlela absorption lona feletseng.
Re lokela ho hlokomela hore e kholoanyane sebaka ya sebakeng se amehileng, le ho feta lithethefatsi tsoela ka Tsamaiso ea tsa bongaka. Ka tsela eo pyatisantimetrovym hlobolisa moriana o "Artrokol" tšoana le 100 g, ketoprfena.
Mora setlolo e sebelisoa, e lokela ho hang-hang hlatsoa matsoho.
O ne a nka gel o lumelloa ho sebelisa ka kopanelo le medicaments tse ling tse nang le ketoprofen (mohlala, ka kopanelo le matlapa a, capsules, rectal suppositories).
The lethal dose palo e kahodimodimo ea moemeli ke mg, 200 ka letsatsi. Ena ke palo ya moriana ha ea itšetleha ka sebōpeho sa meriana.
Ka nako ea 'nete hore phekolo lokela ho ikemisetsa ka motheo oa motho ke ngaka ho ba teng. Leha ho le joalo, re lokela ho hlokomela hore ho sebelisa liniment bakeng sa matsatsi a fetang 10 ka ho latellana e thibetsoe.
litla khoneha lehlakoreng
litla seo mpe li ka etsa hore lithethefatsi "Artrokol" (gel)? Taeo e se buang ka lintho tse latelang litla mpe ea tlhaho:
- bronchospasm, angioedema;
- asthmatic a hlasela, liphetoho anaphylactic ho akarelletsa le makala;
- redness, ho hlohlona, lekhopho, le tuka le ho ruruha ea letlalo;
- bullous phlyctenular eczema le ea nang le bokhoni ba ho jala libakeng tse ling 'me ho ba le eona generalized;
- photosensitivity, bullous kapa ikopanye le dermatitis;
- ho nyekoa ke pelo, Stevens-Johnson lefu, ho hlatsa;
- tsoa mali, liso tsa ka maleng mala, letšollo, lesokolla, pipitlelano;
- Boloetse ba liphio mosebetsi, exacerbation ea renal ho hloleha mofuta foleng, interstitial nephritis le ho hloleha renal.
Ho lokela ho hlokomeloe hore ha ba sebelisa gel "Artrokol" ho ka etsa hore liphetoho tse ling tse lehlakoreng le ka tsamaiso tshilong ya dijo le tsamaiso ea mosese. Le matla liphello tsena itšetlehile ka ka tjhelete e ya lithethefatsi le permeation bokhoni ba motsoako o lona mafolofolo, ho tšoaroa ka eona sebakeng seo boholo, sekhahla le bolelele ba boemo phekolo ea letlalo.
Re ke ke ra bolela hore batho ba hōlileng ba ka ho fetisisa ba tlokotsing ho litla bohloko tsa NSAIDs ka kalafo ya.
Nakong ea bokhachane le ho diabolololo
Nka sebelisa lithethefatsi "Artrokol" (gel) nakong ea bokhachane le kanyeso? Ha ba ntse ba etsa liteko ka litoeba, ho ile ha fumanoa hore ha matlotlo le ha a bake teratogenic le embryotoxic sebetsa ka liphoofolo tse mocha. Leha ho le joalo, re lokela ho hlokomela hore e nyenyane embryotoxic phello e 'nile ha hlokomeloa ka liteko tsa ka mebutlanyana.
Ho tloha ka polokeho ya ketoprofen ka bakhachane ha e so tshehetswa ke lithuto leha e le efe, litsebi li u se ke ua ho kgothaletsa ho sebelisa sesebelisoa sena ho bo-'mè ba moimana.
Hape re lokela ho hlokomela hore ketoprofen le inhibitors tse ling tsa prostaglandin tswakana ka qholotsa toxicity renal, methapo le tsamaiso ea cardiac ya tlhaka ya.
dihlahiswa bola ha matlotlo a fumanoa ka lebese. Ka lebaka lena, ba gel "Artrokol" ha aa lokela ho tsamaisoa ho basali batho ba hlokang tlhokomelo.
lintlha tse hlakileng
Ho lokisetsa "Artrokol" (gel), eo analogs tse boletsoeng ka tlaase, ho e thibetsoe ho sebetsa ho libakeng tse letlalo le liphetoho pathological tse kang lekhopho kapa eczema. E tšoanang e sebetsa ho sebaka seo nang le tšoaetso kapa maqeba bulehileng.
O lokela hape ho qoba lithethefatsi kopana le lera la mucous. Ka mor'a ho sebelisa lithethefatsi o lokela ho hlatsoa matsoho a bona.
sesebelisoa sena ha se a loketse bakeng sa tshebediso ya le dressings occlusive.
Nakong ea kalafo "Artrokolom" le ka libeke tse peli ka mor'a kalafo, ho ke ke tse lakatsehang ho qoba kopana le letlalo ho khanya ea letsatsi ka ho toba.
"Artrokol" (gel): ulasan pelanggan le litokisetso tse tšoanang
Ke analogues ya lithethefatsi ena e kenyeletsa lithethefatsi tse kang "Karmolis-gel", "Indomethacin", "diclofenac", "Remisid", "Vipratoks", "Denebola", "Sepheo sa T", "chondro matla", "Ibuprofen" "Ketonal" le ba bang.
Seo batho ba se buang mabapi le basebelisi ba lithethefatsi? Ba ile ba tlaleha hore gel "Artrokol" e emela e atlehang-ba khahlanong le a hlabang moemeli. Ho sa tšoareng le hantle maemo ao pathological joaloka myalgia, mafu a ea tsamaiso locomotor, mafu a hlabang ea methapong ka, poso-sithabetsang ho ruruha.
The go tlhoka mesola ya meriana ena bakeng sa kopo Link akarelletsa plurality tsa ditlamorao tse bonahatsa maphelong a bona ka mor'a tšebeliso gel. Hangata ka ho fetisisa, bakuli ba a hlokomela ka redness, ho hlohlona, hives, o tukang le ho ruruha ea letlalo, hammoho le ho nyekoa ke pelo, eczema, liso tsa ka maleng mala, letšollo le lesokolla. mosing mong oa lithethefatsi nkoa ke hore e ke ke ea e beuweng ho bakhachane, hammoho le tšebeliso nakong diabolololo.
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